kappa opioid agonistPain Management Peptides

Difelikefalin (Korsuva)

A selective peripherally-restricted kappa opioid receptor agonist. FDA-approved (2021) for pruritus in hemodialysis patients. First-in-class. Does not cross BBB, avoiding central kappa opioid side effects.

anti-pruritickappa-opioid-agonistperipherally-restrictedFDA-approved
3D Structure
3D Structure
679.85 Da
Molecular Weight679.85 Da
FormulaC36H53N7O6
PubChem CID24794466
Lab Tested
No
Harmful Ingredients
0
Contaminants
None
Tested Purity
--
Batch Consistency
No batch data
Mass Spec Profile
Intensity341431522612702m/z680.4
ESI-MS (computed)
Batch Info
Latest Batch
Total Tests0
Unique Vendors0
Vendor Comparison
No vendor data yet
Analysis Summary
Purity Standard
No purity data
Lab Reports
0 reports on file
Summary

A selective peripherally-restricted kappa opioid receptor agonist. FDA-approved (2021) for pruritus in hemodialysis patients. First-in-class. Does not cross BBB, avoiding central kappa opioid side eff…