peptide-drug conjugateOncology Peptides

Melflufen (Pepaxti)

A peptide-drug conjugate with a dipeptide linked to alkylating agent melphalan. FDA-approved (2021, later withdrawn) for relapsed multiple myeloma. Uses aminopeptidase overexpression in cancer cells for selective intracellular drug release.

multiple-myelomaalkylating-agentPDCaminopeptidase-targeted
3D Structure
3D Structure
498.4 Da
63 atoms
Molecular Weight498.4 Da
FormulaC24H30Cl2FN3O3
PubChem CID9935639
Lab Tested
No
Harmful Ingredients
0
Contaminants
None
Tested Purity
--
Batch Consistency
No batch data
Mass Spec Profile
Intensity250317385453520m/z498.2
ESI-MS (computed)
Batch Info
Latest Batch
Total Tests0
Unique Vendors0
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Analysis Summary
Purity Standard
No purity data
Lab Reports
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Summary

A peptide-drug conjugate with a dipeptide linked to alkylating agent melphalan. FDA-approved (2021, later withdrawn) for relapsed multiple myeloma. Uses aminopeptidase overexpression in cancer cells f…